TargetMol

GRL0617

Product Code:
 
TAR-T11464
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11464-1mg1mg£95.00
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TAR-T11464-5mg5mg£128.00
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TAR-T11464-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T11464-10mg10mg£161.00
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TAR-T11464-25mg25mg£230.00
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TAR-T11464-50mg50mg£349.00
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TAR-T11464-100mg100mg£516.00
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TAR-T11464-500mg500mg£1,018.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM).
CAS:
1093070-16-6
Formula:
C20H20N2O
Molecular Weight:
304.393
Pathway:
Cell Cycle/Checkpoint; Microbiology/Virology; Ubiquitination; DNA Damage/DNA Repair
Purity:
0.9977
SMILES:
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc2ccccc12
Target:
SARS-CoV; DUB

References

1. Ratia K, et al. A noncovalent class of papain-like protease/deubiquitinase inhibitors blocks SARS virus replication. Proc Natl Acad Sci U S A. 2008 Oct 21;105(42):16119-24.