TargetMol

Epelsiban

Product Code:
 
TAR-T11502
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11502-5mg5mg£1,171.00
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TAR-T11502-50mg50mg£2,303.00
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Quantity:
TAR-T11502-100mg100mg£3,042.00
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This product comes from: United States.
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Further Information

Bioactivity:
Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).
CAS:
872599-83-2
Formula:
C30H38N4O4
Molecular Weight:
518.658
Purity:
0.98
SMILES:
[H][C@]1([C@@H](C)CC)N([C@@H](C(=O)N2CCOCC2)c2ccc(C)nc2C)C(=O)[C@H](NC1=O)C1Cc2ccccc2C1

References

1. Borthwick AD, et al. Pyridyl-2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists: synthesis, pharmacokinetics, and in vivo potency. J Med Chem. 2012 Jan 26;55(2):783-96.