TargetMol

HDAC-IN-4

Product Code:
 
TAR-T11542
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
HDAC-IN-4 is a selective HDAC6 and HDAC10 inhibitor (pIC50s: 7.2 and 6.8 in BRET assay) with antitumoral activity.
CAS:
1252003-13-6
Formula:
C20H21N3O2
Molecular Weight:
335.407
Pathway:
DNA Damage/DNA Repair; Chromatin/Epigenetic
Purity:
0.98
SMILES:
CN1CCc2c(C1)n(Cc1ccc(cc1)C(=O)NO)c1ccccc21
Target:
HDAC

References

1. G?raldy M, et al. Selective Inhibition of Histone Deacetylase 10: Hydrogen Bonding to the Gatekeeper Residue is Implicated. J Med Chem. 2019 May 9;62(9):4426-4443.