TargetMol

JAK2-IN-4

Product Code:
 
TAR-T11708
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T11708-5mg5mg£1,091.00
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TAR-T11708-50mg50mg£2,143.00
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Quantity:
TAR-T11708-100mg100mg£2,801.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
JAK2-IN-4 is a selective JAK2/JAK3 inhibitor, with IC50 values of 0.7 nM and 23.2 nM for JAK2 and JAK3, respectively.
CAS:
1438284-00-4
Formula:
C23H27N5O4S
Molecular Weight:
469.56
Pathway:
Angiogenesis; JAK/STAT signaling; Stem Cells; Chromatin/Epigenetic
Purity:
0.98
SMILES:
Cc1cnc(Nc2ccc(cc2)N2CCOCC2)nc1-c1cc2CN(CCc2o1)S(C)(=O)=O
Target:
JAK

References

1. Wang Y, et al. Identification of 4-(2-furanyl)pyrimidin-2-amines as Janus kinase 2 inhibitors. Bioorg Med Chem. 2017 Jan 1;25(1):75-83.