TargetMol

Lesopitron dihydrochloride

Product Code:
 
TAR-T11839
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11839-5mg5mg£850.00
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TAR-T11839-50mg50mg£1,661.00
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TAR-T11839-100mg100mg£2,079.00
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Further Information

Bioactivity:
Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.
CAS:
132449-89-9
Formula:
C15H23Cl3N6
Molecular Weight:
393.74
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
Cl.Cl.Clc1cnn(CCCCN2CCN(CC2)c2ncccn2)c1
Target:
5-HT Receptor

References

1. Haj-Dahmane S, et al. Interactions of Lesopitron (E-4424) with central 5-HT1A receptors: in vitro and in vivo studies in the rat. Eur J Pharmacol. 1994 Apr 1;255(1-3):185-96. 2. Ballar?n M, et al. Effect of acute administration of the 5-HT1A receptor ligand, Lesopitron, on rat cortical 5-HT and dopamine turnover. Br J Pharmacol. 1994 Oct;113(2):425-30.