TargetMol

McN5691

Product Code:
 
TAR-T11979
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11979-5mg5mg£850.00
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TAR-T11979-50mg50mg£1,661.00
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Quantity:
TAR-T11979-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
McN5691 is a voltage sensitive calcium channel blocker.
CAS:
99254-95-2
Formula:
C30H35NO3
Molecular Weight:
457.614
Pathway:
Membrane transporter/Ion channel; Metabolism
Purity:
0.98
SMILES:
COc1ccc(C#Cc2ccccc2)c(CCC(C)N(C)CCc2ccc(OC)c(OC)c2)c1
Target:
Calcium Channel

References

1. Flaim SF, et al. Structurally novel antihypertensive compound, McN-5691, is a calcium channel blocker in vascular smooth muscle. J Pharmacol Exp Ther. 1991 Jan;256(1):279-88. 2. Wu WN, et al. Excretion and metabolism of the antihypertensive agent, RWJ-26240 (McN-5691) in dogs. Drug Metab Dispos. 1998 Feb;26(2):115-25. 3. Flaim SF, et al. Effects of the novel calcium channel blocker, McN-5691, on cardiocirculatory dynamics and cardiac output distribution in conscious spontaneously hypertensive rat. J Cardiovasc Pharmacol. 1988 Apr;11(4):489-500.