TargetMol

PARP/PI3K-IN-1

Product Code:
 
TAR-T12365
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12365-5mg5mg£404.00
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TAR-T12365-50mg50mg£1,661.00
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Quantity:
TAR-T12365-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PARP/PI3K-IN-1 is a potent inhibitor of PARP/PI3K(pIC50 values of 8.22).
CAS:
2337386-47-5
Formula:
C33H28F4N8O3
Molecular Weight:
660.634
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
Nc1cc(c(cn1)-c1nc2CN(CCc2c(n1)N1CCOCC1)C(=O)c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F)C(F)(F)F
Target:
PI3K

References

1. Wang J, et al.Discovery of Novel Dual Poly(ADP-ribose)polymerase and Phosphoinositide 3-Kinase Inhibitors as a Promising Strategy for Cancer Therapy.J Med Chem. 2020 Jan 9;63(1):122-139.