TargetMol

PI3kδ inhibitor 1

Product Code:
 
TAR-T12463
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12463-5mg5mg£1,492.00
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TAR-T12463-50mg50mg£2,946.00
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Quantity:
TAR-T12463-100mg100mg£4,006.00
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This product comes from: United States.
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Further Information

Bioactivity:
PI3kδ inhibitor 1 is a selective inhibitor of PI3Kδ (IC50 of 3.8 nM).
CAS:
1332075-63-4
Formula:
C28H33FN6O2
Molecular Weight:
504.61
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
CC(C)(O)C1CCN(Cc2ccc3nc(nc(N4CCOCC4)c3n2)-c2c(F)ccc3[nH]ccc23)CC1
Target:
PI3K

References

1. Sutherlin DP, et al. Potent and selective inhibitors of PI3K?: obtaining isoform selectivity from the affinity pocket and tryptophan shelf. Bioorg Med Chem Lett. 2012 Jul 1;22(13):4296-302.