TargetMol

Pinacidil

Product Code:
 
TAR-T12478L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T12478L-5mg5mg£104.00
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TAR-T12478L-1mL1 mL * 10 mM (in DMSO)£107.00
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TAR-T12478L-10mg10mg£117.00
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TAR-T12478L-25mg25mg£148.00
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Quantity:
TAR-T12478L-50mg50mg£203.00
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This product comes from: United States.
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Further Information

Bioactivity:
Pinardil (P-1134, S-1230) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and peripheral resistance and producing fluid retention.
CAS:
60560-33-0
Formula:
C13H19N5
Molecular Weight:
245.33
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CC(C)(C)C(N/C(NC1=CC=NC=C1)=N/C#N)C
Target:
Potassium Channel

References

1. Friedel HA, Brogden RN. Pinacidil. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in the treatment of hypertension. Drugs. 1990 Jun;39(6):929-67. Review. PubMed PMID: 2196168. 2. Ahnfelt-R?nne I. Pinacidil. Preclinical investigations. Drugs. 1988;36 Suppl 7:4-9. Review. PubMed PMID: 3076134. 3. Cohen ML, Kurz KD. Pinacidil-induced vascular relaxation: comparison to other vasodilators and to classical mechanisms of vasodilation. J Cardiovasc Pharmacol. 1988;12 Suppl 2:S5-9. PubMed PMID: 2466179. 4. Zushida K, Onodera K, Kamei J. Effect of diabetes on pinacidil-induced antinociception in mice. Eur J Pharmacol. 2002 Oct 25;453(2-3):209-15. PubMed PMID: 12398906.