TargetMol

PROTAC BRD9 Degrader-1

Product Code:
 
TAR-T12560
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12560-5mg5mg£659.00
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Quantity:
TAR-T12560-10mg10mg£1,050.00
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This product comes from: United States.
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Further Information

Bioactivity:
PROTAC BRD9 Degrader-1 is a lead PROTAC BRD9 chemical degrader with IC50 of 13.5 nM.
CAS:
2097971-01-0
Formula:
C42H45N7O12S2
Molecular Weight:
903.98
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
COc1cc(ccc1OCC(=O)NCCCCNC(=O)COc1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12)-c1cn(C)c(=O)c2cc(sc12)C(=N)NC1CCS(=O)(=O)CC1
Target:
Epigenetic Reader Domain

References

1. Remillard D, et al. Degradation of the BAF Complex Factor BRD9 by Heterobifunctional Ligands. Angew Chem Int Ed Engl. 2017 May 15;56(21):5738-5743.