TargetMol

ROS 234 dioxalate

Product Code:
 
TAR-T12756
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12756-5mg5mg£850.00
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Quantity:
TAR-T12756-50mg50mg£1,661.00
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Quantity:
TAR-T12756-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)
CAS:
1781941-93-2
Formula:
C17H19N5O8
Molecular Weight:
421.366
Pathway:
Neuroscience; Immunology/Inflammation; GPCR/G Protein
Purity:
0.98
SMILES:
OC(=O)C(O)=O.OC(=O)C(O)=O.C(CNc1nc2ccccc2[nH]1)Cc1cnc[nH]1
Target:
Histamine Receptor

References

1. Ballabeni V, et al. CNS access of selected H3-antagonists: ex vivo binding study in rats. Inflamm Res. 2002 Apr;51 Suppl 1:S55-6. 2. Mor M, et al. Synthesis, biological activity, QSAR and QSPR study of 2-aminobenzimidazole derivatives as potent H3-antagonists. Bioorg Med Chem. 2004 Feb 15;12(4):663-74.