TargetMol

SA57

Product Code:
 
TAR-T12826
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12826-5mg5mg£850.00
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Quantity:
TAR-T12826-50mg50mg£1,661.00
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Quantity:
TAR-T12826-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
CAS:
1346169-63-8
Formula:
C17H23ClN2O3
Molecular Weight:
338.83
Pathway:
Metabolism; Neuroscience
Purity:
0.98
SMILES:
CNC(=O)COC(=O)N1CCC(CCc2ccc(Cl)cc2)CC1
Target:
FAAH

References

1. Niphakis MJ, et al. O-hydroxyacetamide carbamates as a highly potent and selective class of endocannabinoid hydrolase inhibitors. ACS Chem Neurosci. 2012 May 16;3(5):418-26. 2. Owens RA, et al. Discriminative Stimulus Properties of the Endocannabinoid Catabolic Enzyme Inhibitor SA-57 in Mice. J Pharmacol Exp Ther. 2016 Aug;358(2):306-14.