TargetMol

SGLT inhibitor-1

Product Code:
 
TAR-T12893
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12893-5mg5mg£1,412.00
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TAR-T12893-50mg50mg£2,785.00
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Quantity:
TAR-T12893-100mg100mg£3,765.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s of 43 nM and 9 nM, respectively).
CAS:
2247314-23-2
Formula:
C24H27FO8
Molecular Weight:
462.47
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
COc1c2CCOc2c(Cc2ccc3OCCOc3c2)cc1[C@@H]1O[C@H](CO)[C@@H](F)[C@H](O)[C@H]1O
Target:
SGLT

References

1. Xu G? et al. Design, synthesis and biological evaluation of (2S,3R,4R,5S,6R)-5-fluoro-6-(hydroxymethyl)-2-aryltetrahydro-2H-pyran-3,4-diols as potent and orally active SGLT dual inhibitors. Bioorg Med Chem Lett. 2018 Nov 15;28(21):3446-3453.