TargetMol

SMYD3-IN-1

Product Code:
 
TAR-T12940
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12940-5mg5mg£470.00
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TAR-T12940-50mg50mg£1,982.00
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Quantity:
TAR-T12940-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
SMYD3-IN-1 is an irreversible and selective SMYD3 (SET and MYND domain containing 3) inhibitor(IC50 of 11.7 nM).
CAS:
2095160-79-3
Formula:
C28H31ClN4O3
Molecular Weight:
507.03
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
CCCOC(=O)N1CCN(C[C@H]1C)C(=O)c1ccc2c(Cl)cc(nc2c1)-c1ccc(cc1)C1(N)CC1
Target:
Histone Methyltransferase

References

1. Huang C, et al. Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3. ACS Med Chem Lett. 2019 May 23;10(6):978-984.