TargetMol

S2101

Product Code:
 
TAR-T13052
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
S 2101 is an inhibitor of lysine-specific demethylase 1 (LSD1)(IC50 of 0.99 μM, Ki of 0.61 μM and Kinact/Ki of 4560 M/s).
CAS:
1239262-36-2
Formula:
C16H16ClF2NO
Molecular Weight:
311.76
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
Cl.N[C@@H]1C[C@H]1c1cc(F)cc(F)c1OCc1ccccc1
Target:
Histone Demethylase

References

1. Mimasu S, et al. Structurally designed trans-2-phenylcyclopropylamine derivatives potently inhibit histone demethylase LSD1/KDM1 . Biochemistry. 2010 Aug 3;49(30):6494-503.