TargetMol

UbcH5c-IN-1

Product Code:
 
TAR-T13242
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13242-5mg5mg£850.00
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Quantity:
TAR-T13242-50mg50mg£1,661.00
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Quantity:
TAR-T13242-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
UbcH5c-IN-1 is a selective small-molecule Ubiquitin-conjugating enzyme UbcH5c inhibitor (Kd: 283 nM for E2 UbcH5c-IN-1 by covalent binding with Cys85).
CAS:
2123480-72-6
Formula:
C22H21BrO3
Molecular Weight:
413.311
Purity:
0.98
SMILES:
Cc1cc(OCc2ccccc2Br)c(C)c2[C@@H]3OC(=O)C(=C)[C@@H]3CCc12

References

1. Chen H, et al. Discovery of Potent Small-Molecule Inhibitors of Ubiquitin-Conjugating Enzyme UbcH5c from ?-Santonin Derivatives. J Med Chem. 2017 Aug 24;60(16):6828-6852.