TargetMol

VU591 hydrochloride

Product Code:
 
TAR-T13320
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
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CodeSizePrice
TAR-T13320-1mg1mg£193.00
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TAR-T13320-5mg5mg£370.00
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TAR-T13320-1mL1 mL * 10 mM (in DMSO)£412.00
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TAR-T13320-10mg10mg£519.00
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TAR-T13320-25mg25mg£791.00
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TAR-T13320-50mg50mg£1,058.00
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TAR-T13320-100mg100mg£1,404.00
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TAR-T13320-500mg500mg£2,737.00
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Further Information

Bioactivity:
VU591 hydrochloride is a selective renal outer medullary potassium channel (Kir1.1, ROMK) antagonist (IC50?0.24 μM). Thought to block the intracellular pore of the Kir1.1 channel. Exhibits no effect on Kir7.1 at concentrations up to 10 μM; does not inhibit Kir2.1, Kir2.3 or Kir4.1. Displays similar potency to VU 590
CAS:
1315380-70-1
Formula:
C16H13ClN6O5
Molecular Weight:
404.77
Pathway:
Membrane transporter/Ion channel
Purity:
0.9995
SMILES:
Cl.[O-][N+](=O)c1ccc2nc(COCc3nc4ccc(cc4[nH]3)[N+]([O-])=O)[nH]c2c1
Target:
Potassium Channel

References

1. Bhave G, et al. Development of a selective small-molecule inhibitor of Kir1.1, the renal outer medullary potassium channel. Mol Pharmacol. 2011 Jan;79(1):42-50.