TargetMol

JTE-013

Product Code:
 
TAR-T15629
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15629-5mg5mg£127.00
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TAR-T15629-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T15629-10mg10mg£152.00
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TAR-T15629-25mg25mg£250.00
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TAR-T15629-50mg50mg£340.00
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Further Information

Bioactivity:
JTE-013 is an effective and specific antagonist of S1P2. JTE-013 suppresses the specific binding of radiolabeled S1P to human and rat S1P2 (IC50s: 17 nM and 22 nM, respectively).
CAS:
383150-41-2
Formula:
C17H19Cl2N7O
Molecular Weight:
408.29
Pathway:
Apoptosis; GPCR/G Protein
Purity:
0.9887
SMILES:
CC(C)c1cc(NNC(=O)Nc2cc(Cl)nc(Cl)c2)nc2n(C)nc(C)c12
Target:
Apoptosis; S1P Receptor; LPL Receptor

References

1. Li MH, et al. Antitumor Activity of a Novel Sphingosine-1-Phosphate 2 Antagonist, AB1, in Neuroblastoma. J Pharmacol Exp Ther. 2015 Sep;354(3):261-8.