TargetMol

Kelatorphan

Product Code:
 
TAR-T15652
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15652-5mg5mg£617.00
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Quantity:
TAR-T15652-50mg50mg£1,982.00
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Quantity:
TAR-T15652-100mg100mg£2,560.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Kelatorphan is an enkephalin degrading enzyme full inhibitor.
CAS:
92175-57-0
Formula:
C14H18N2O5
Molecular Weight:
294.307
Purity:
0.98
SMILES:
C[C@H](NC(=O)[C@@H](CC(=O)NO)Cc1ccccc1)C(O)=O

References

1. Waksman G, et al. Kelatorphan: a full inhibitor of enkephalin degrading enzymes. Biochemical and pharmacological properties, regional distribution of enkephalinase in rat brain by use of a tritiated derivative. Neuropeptides. 1985 Feb;5(4-6):529-32. 2. Waksman G, et al. In vitro and in vivo effects of kelatorphan on enkephalin metabolism in rodent brain. Eur J Pharmacol. 1985 Nov 5;117(2):233-43. 3. Boudinot E, et al. Effects of the potent analgesic enkephalin-catabolizing enzyme inhibitors RB101 and kelatorphan on respiration. Pain. 2001 Feb 1;90(1-2):7-13.