TargetMol

LPA1 receptor antagonist 1

Product Code:
 
TAR-T15785
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15785-5mg5mg£1,010.00
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TAR-T15785-50mg50mg£1,982.00
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TAR-T15785-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
LPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist (IC50: 25 nM).
CAS:
1396006-71-5
Formula:
C28H26N4O4
Molecular Weight:
482.54
Pathway:
Immunology/Inflammation
Purity:
0.98
SMILES:
C[C@@H](OC(=O)Nc1c(C)nnn1-c1ccc(cc1)-c1ccc(cc1)C1(CC1)C(O)=O)c1ccccc1
Target:
TLR

References

1. Qian Y, et al. Discovery of highly selective and orally active lysophosphatidic acid receptor-1 antagonists with potent activity on human lung fibroblasts. J Med Chem. 2012 Sep 13;55(17):7920-39.