TargetMol

Pelubiprofen

Product Code:
 
TAR-T16464
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16464-5mg5mg£850.00
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Further Information

Bioactivity:
Pelubiprofen inhibits COX activity and the transforming growth factor-β activated kinase 1-IκB kinase β-NF-κB pathway. It also has significant anti-inflammatory and analgesic effects. Pelubiprofen is an orally active and non-steroidal anti-inflammatory drug and is a member of the 2-arylpropionic acid family and has relatively selective effects on COX-2 activity .
CAS:
69956-77-0
Formula:
C16H18O3
Molecular Weight:
258.317
Pathway:
Neuroscience; Immunology/Inflammation
Purity:
0.98
SMILES:
CC(C(O)=O)c1ccc(C=C2/CCCCC2=O)cc1
Target:
COX

References

1. Choi IA, Baek HJ, et al. Comparison of the efficacy and safety profiles of a pelubiprofen versus celecoxib in patients with rheumatoid arthritis: a 6-week, multicenter, randomized, double-blind, phase III, non-inferiority clinical trial. BMC Musculoskelet Disord. 2014 Nov 18;15:375.