TargetMol

PF-05241328

Product Code:
 
TAR-T16487
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16487-5mg5mg£277.00
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TAR-T16487-50mg50mg£962.00
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TAR-T16487-100mg100mg£1,508.00
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This product comes from: United States.
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Further Information

Bioactivity:
PF-05241328 is an effective and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (IC50: 31 nM).
CAS:
1387633-03-5
Formula:
C19H21ClN4O4S
Molecular Weight:
436.91
Purity:
0.98
SMILES:
CC(C)COc1ncc(cc1Cl)-n1nc(C)c2cc(ccc12)C(=O)NS(C)(=O)=O

References

1. Jones HM, et al. Clinical Micro-Dose Studies to Explore the Human Pharmacokinetics of Four Selective Inhibitors of Human Nav1.7 Voltage-Dependent Sodium Channels. Clin Pharmacokinet. 2016 Jul;55(7):875-887.