TargetMol

PF-06795071

Product Code:
 
TAR-T16496
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16496-5mg5mg£1,332.00
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Quantity:
TAR-T16496-50mg50mg£2,625.00
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Quantity:
TAR-T16496-100mg100mg£3,524.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).
CAS:
2075629-81-9
Formula:
C18H17F4N3O3
Molecular Weight:
399.346
Pathway:
Metabolism
Purity:
0.98
SMILES:
[H][C@@]12CN(C[C@]1([H])[C@H]2c1ccn(n1)-c1ccc(F)cc1)C(=O)O[C@H](CO)C(F)(F)F
Target:
Lipase

References

1. McAllister LA, et al. Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation. J Med Chem. 2018 Apr 12;61(7):3008-3026.