TargetMol

XMD8-92

Product Code:
 
TAR-T1843
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T1843-5mg5mg£109.00
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TAR-T1843-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T1843-10mg10mg£125.00
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TAR-T1843-25mg25mg£177.00
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TAR-T1843-50mg50mg£269.00
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Quantity:
TAR-T1843-100mg100mg£402.00
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Further Information

Bioactivity:
XMD8-92 is an effective and specific BMK1/ERK5 inhibitor (Kd: 80 nM).
CAS:
1234480-50-2
Formula:
C26H30N6O3
Molecular Weight:
474.565
Pathway:
Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK
Purity:
0.9819
SMILES:
CCOc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCC(O)CC1
Target:
ERK; BMI-1; Epigenetic Reader Domain

References

1. Yang Q, et al. Cancer Cell. 2010, 18(3), 258-267. 2. Dong H, et al. Pharm Biol. 2013. doi:10.3109/13880209. 3. Sureban SM, et al. Cancer Lett. 2014 , 351(1), 151-161.