TargetMol

GSK3787

Product Code:
 
TAR-T1941
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T1941-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T1941-5mg5mg£111.00
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TAR-T1941-10mg10mg£134.00
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TAR-T1941-25mg25mg£217.00
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TAR-T1941-50mg50mg£332.00
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TAR-T1941-100mg100mg£511.00
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TAR-T1941-500mg500mg£1,010.00
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This product comes from: United States.
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Further Information

Bioactivity:
GSK3787 is a specific and irreversible PPARδ inhibitor?pIC50= 6.6?.
CAS:
188591-46-0
Formula:
C15H12ClF3N2O3S
Molecular Weight:
392.78
Pathway:
Metabolism; DNA Damage/DNA Repair
Purity:
0.9805
SMILES:
FC(F)(F)c1ccc(nc1)S(=O)(=O)CCNC(=O)c1ccc(Cl)cc1
Target:
PPAR

References

1. Shearer BG, et al. J Med Chem, 2010, 53(4), 1857-1861. 2. Palkar PS, et al. Mol Pharmacol, 2010, 78(3) 419-430. 3. Brown PJ, et al. Chem Biol, 1997, 4(12), 909-918.