TargetMol

PD153035

Product Code:
 
TAR-T2041
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2041-5mg5mg£102.00
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Quantity:
TAR-T2041-1mL1 mL * 10 mM (in DMSO)£116.00
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Quantity:
TAR-T2041-10mg10mg£117.00
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TAR-T2041-25mg25mg£168.00
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Quantity:
TAR-T2041-50mg50mg£251.00
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Quantity:
TAR-T2041-100mg100mg£386.00
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Quantity:
TAR-T2041-200mg200mg£544.00
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Quantity:
TAR-T2041-500mg500mg£812.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
PD153035 hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free assays); little inhibitory against FGFR, PGDFR, InsR, CSF-1 and Src.
CAS:
153436-54-5
Formula:
C16H14BrN3O2
Molecular Weight:
360.211
Pathway:
JAK/STAT signaling; Angiogenesis; Tyrosine Kinase/Adaptors
Purity:
0.9931
SMILES:
COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OC
Target:
EGFR

References

1. Fry DW, et al. Science. 1994, 265(5175), 1093-1095.