TargetMol

AS-041164

Product Code:
 
TAR-T21938
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T21938-5mg5mg£102.00
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TAR-T21938-1mL1 mL * 10 mM (in DMSO)£105.00
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TAR-T21938-10mg10mg£122.00
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TAR-T21938-25mg25mg£169.00
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TAR-T21938-50mg50mg£253.00
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TAR-T21938-100mg100mg£364.00
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TAR-T21938-200mg200mg£458.00
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TAR-T21938-500mg500mg£704.00
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Further Information

Bioactivity:
AS-041164 is a selective and orally active PI3Kγ isoform inhibitor(IC50 of 70 nM), and shows less activity against PI3Kα, PI3Kβ, and PI3Kδ (IC50s of 240 nM, 1.45 μM, and 1.70 μM, respectively). It has anti-inflammatory effects.
CAS:
6318-41-8
Formula:
C11H7NO4S
Molecular Weight:
249.24
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.9959
SMILES:
O=C1NC(=O)C(S1)=Cc1ccc2OCOc2c1
Target:
PI3K

References

1. Chiara Ferrandi, et al. Phosphoinositide 3-kinase gamma inhibition plays a crucial role in early steps of inflammation by blocking neutrophil recruitment. J Pharmacol Exp Ther. 2007 Sep;322(3):923-30.