TargetMol

BGT1-IN-9

Product Code:
 
TAR-T23787
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T23787-5mg5mg£850.00
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Quantity:
TAR-T23787-50mg50mg£1,661.00
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Quantity:
TAR-T23787-100mg100mg£2,079.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
BGT1-IN-9 is an M1 muscarinic agonist.
CAS:
185444-92-2
Formula:
C5H10ClN3O2
Molecular Weight:
179.6
Purity:
0.98
SMILES:
Cl.NC1=NCC(CN1)C(O)=O

References

1. Al-Khawaja A, Haugaard AS, Marek A, L?ffler R, Thiesen L, Santiveri M, Damgaard M, Bundgaard C, Fr?lund B, Wellendorph P. Pharmacological Characterization of [(3)H]ATPCA as a Substrate for Studying the Functional Role of the Betaine/GABA Transporter 1 and the Creatine Transporter. ACS Chem Neurosci. 2018 Mar 21;9(3):545-554. doi: 10.1021/acschemneuro.7b00351. Epub 2017 Nov 22. PubMed PMID: 29131576. 2. Al-Khawaja A, Petersen JG, Damgaard M, Jensen MH, Vogensen SB, Lie ME, Kragholm B, Br?uner-Osborne H, Clausen RP, Fr?lund B, Wellendorph P. Pharmacological identification of a guanidine-containing ?-alanine analogue with low micromolar potency and selectivity for the betaine/GABA transporter 1 (BGT1). Neurochem Res. 2014 Oct;39(10):1988-96. doi: 10.1007/s11064-014-1336-9. Epub 2014 May 23. PubMed PMID: 24852577. 3. Su?ol C, Babot Z, Crist?fol R, Sonnewald U, Waagepetersen HS, Schousboe A. A possible role of the non-GAT1 GABA transporters in transfer of GABA from GABAergic to glutamatergic neurons in mouse cerebellar neuronal cultures. Neurochem Res. 2010 Sep;35(9):1384-90. doi: 10.1007/s11064-010-0196-1. Epub 2010 May 30. PubMed PMID: 20512624. 4. Moeckel GW, Zhang L, Fogo AB, Hao CM, Pozzi A, Breyer MD. COX2 activity promotes organic osmolyte accumulation and adaptation of renal medullary interstitial cells to hypertonic stress. J Biol Chem. 2003 May 23;278(21):19352-7. Epub 2003 Mar 9. PubMed PMID: 12637551.