TargetMol

D 595

Product Code:
 
TAR-T23932
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T23932-5mg5mg£850.00
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Quantity:
TAR-T23932-50mg50mg£1,661.00
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Quantity:
TAR-T23932-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
D595 is a phenethylamine-type calcium channel blocker. The most potent phenylethylamine with respect to negative inotropy was D595 (EC50: 794 nmol/l).
CAS:
16740-29-7
Formula:
C25H32Cl2N2O2
Molecular Weight:
463.44
Purity:
0.98
SMILES:
COc1ccc(CCN(C)CCCC(C#N)(C(C)C)c2ccc(Cl)c(Cl)c2)cc1OC

References

1. Clark JM, Brooks MW. Role of ion channels and intraterminal calcium homeostasis in the action of deltamethrin at presynaptic nerve terminals. Biochem Pharmacol. 1989 Jul 15;38(14):2233-45. PubMed PMID: 2546560. 2. Goll A, Glossmann H, Mannhold R. Correlation between the negative inotropic potency and binding parameters of 1,4-dihydropyridine and phenylalkylamine calcium channel blockers in cat heart. Naunyn Schmiedebergs Arch Pharmacol. 1986 Nov;334(3):303-12. PubMed PMID: 3027587.