TargetMol

DAT 582

Product Code:
 
TAR-T23965
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T23965-5mg5mg£930.00
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Quantity:
TAR-T23965-50mg50mg£1,821.00
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Quantity:
TAR-T23965-100mg100mg£2,319.00
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This product comes from: United States.
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Further Information

Bioactivity:
DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agent
CAS:
141034-42-6
Formula:
C22H29Cl2N5O
Molecular Weight:
450.41
Purity:
0.98
SMILES:
O=C(C1=NNC2=C1C=CC=C2)N[C@H]3CN(CC4=CC=CC(C)=C4)CCN(C)C3.[H]Cl.[H]Cl

References

1. Meyer O, Hoffmann T, Aslan T, Ahrens N, Kiesewetter H, Salama A. Diclofenac-induced antibodies against RBCs and platelets: two case reports and a concise review. Transfusion. 2003 Mar;43(3):345-9. Review. PubMed PMID: 12675720. 2. Kato S, Fujiwara I, Yoshida N. Nitrogen-containing heteroalicycles with serotonin receptor binding affinity: development of gastroprokinetic and antiemetic agents. Med Res Rev. 1999 Jan;19(1):25-73. Review. PubMed PMID: 9918193. 3. Newberry NR, Sprosen TS, Watkins CJ, Leslie RA, Grahame-Smith DG. AS-5370 potently antagonizes 5-HT3 receptor-mediated responses on NG108-15 cells and on the rat vagus. Eur J Pharmacol. 1992 Aug 14;219(1):135-40. PubMed PMID: 1397040. 4. Yoshida N, Omoya H, Kato S, Ito T. 5-HT3 receptor antagonist effects of DAT-582, (R) enantiomer of AS-5370. Eur J Pharmacol. 1992 Jun 17;216(3):435-40. PubMed PMID: 1425931.