TargetMol

Deltazinone

Product Code:
 
TAR-T23977
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T23977-5mg5mg£850.00
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Quantity:
TAR-T23977-50mg50mg£1,661.00
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Quantity:
TAR-T23977-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Deltazinone is a selective PDEδ inhibitor. Deltazinone exhibits less unspecific cytotoxicity and demonstrates a high correlation with the phenotypic effect of PDEδ knockdown in a set of human pancreatic cancer cell lines.
CAS:
894554-89-3
Formula:
C27H31N5O2
Molecular Weight:
457.578
Purity:
0.98
SMILES:
CC(CNC(=O)CCCn1nc(C)c2c(C)n(nc2c1=O)-c1ccc(C)cc1)c1ccccc1

References

1. Papke B, Murarka S, Vogel HA, Mart?n-Gago P, Kovacevic M, Truxius DC, Fansa EK, Ismail S, Zimmermann G, Heinelt K, Schultz-Fademrecht C, Al Saabi A, Baumann M, Nussbaumer P, Wittinghofer A, Waldmann H, Bastiaens PI. Identification of pyrazolopyridazinones as PDE? inhibitors. Nat Commun. 2016 Apr 20;7:11360. doi: 10.1038/ncomms11360. PubMed PMID: 27094677; PubMed Central PMCID: PMC4843002.