TargetMol

HDAC3-IN-T247

Product Code:
 
TAR-T24131
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T24131-50mg50mg£962.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T24131-100mg100mg£1,364.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
HDAC3-IN-T247 is a potent and selective HDAC3 inhibitor that acts by increasing NF-κB acetylation. It also activating HIV gene expression in latent HIV-infected cells.
CAS:
1451042-18-4
Formula:
C21H19N5OS
Molecular Weight:
389.48
Purity:
0.98
SMILES:
Nc1ccccc1NC(=O)c1ccc(cc1)-c1cn(CCc2ccsc2)nn1

References

1. Suzuki T, Kasuya Y, Itoh Y, Ota Y, Zhan P, Asamitsu K, Nakagawa H, Okamoto T, Miyata N. Identification of highly selective and potent histone deacetylase 3 inhibitors using click chemistry-based combinatorial fragment assembly. PLoS One. 2013 Jul 16;8(7):e68669. doi: 10.1371/journal.pone.0068669. Print 2013. PubMed PMID: 23874714; PubMed Central PMCID: PMC3713009.