TargetMol

L 368935

Product Code:
 
TAR-T24293
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24293-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T24293-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T24293-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
L 368935 is an antagonist of the cholecystokinin receptor.
CAS:
145878-31-5
Formula:
C27H26N8O2
Molecular Weight:
494.559
Purity:
0.98
SMILES:
CC(C)CN1c2ccccc2C(=N[C@@H](NC(=O)Nc2cccc(c2)-c2nnn[nH]2)C1=O)c1ccccc1

References

1. Patel S, Chapman KL, Smith AJ, Heald A, Freedman SB. Use of ex vivo binding to estimate brain penetration and central activity of CCK-B antagonists. Ann N Y Acad Sci. 1994 Mar 23;713:360-3. PubMed PMID: 8185188. 2. Pedersen K, Nielsen FC, Rehfeld JF. Regulation of the human cholecystokinin gene. Ann N Y Acad Sci. 1994 Mar 23;713:321-3. PubMed PMID: 8185176. 3. Patel S, Chapman KL, Heald A, Smith AJ, Freedman SB. Measurement of central nervous system activity of systemically administered CCKB receptor antagonists by ex vivo binding. Eur J Pharmacol. 1994 Mar 3;253(3):237-44. PubMed PMID: 8200418.