TargetMol

GSK2801

Product Code:
 
TAR-T2436
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T2436-1mg1mg£95.00
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TAR-T2436-2mg2mg£102.00
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TAR-T2436-5mg5mg£119.00
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TAR-T2436-1mL1 mL * 10 mM (in DMSO)£121.00
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TAR-T2436-10mg10mg£134.00
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TAR-T2436-25mg25mg£215.00
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TAR-T2436-50mg50mg£330.00
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TAR-T2436-100mg100mg£503.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK2801 is an effective, specific and cell active acetyl-lysine competitive inhibitor of BAZ2A(Kd: 136 nM) and BAZ2B(Kd: 257 nM) bromodomains.
CAS:
1619994-68-1
Formula:
C20H21NO4S
Molecular Weight:
371.45
Pathway:
Apoptosis; Chromatin/Epigenetic
Purity:
0.9988
SMILES:
CCCOc1ccn2c(cc(-c3ccccc3S(C)(=O)=O)c2c1)C(C)=O
Target:
Apoptosis; Epigenetic Reader Domain

References

1. Chen P, et al. 2015. DOI: 10.1021/acs.jmedchem.5b00209