TargetMol

CPI203

Product Code:
 
TAR-T2442
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2442-1mL1 mL * 10 mM (in DMSO)£111.00
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TAR-T2442-5mg5mg£111.00
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TAR-T2442-10mg10mg£131.00
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TAR-T2442-25mg25mg£167.00
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TAR-T2442-50mg50mg£248.00
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TAR-T2442-100mg100mg£390.00
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This product comes from: United States.
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Further Information

Bioactivity:
CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).
CAS:
202591-23-9
Formula:
C19H18ClN5OS
Molecular Weight:
399.9
Pathway:
Chromatin/Epigenetic
Purity:
0.9913
SMILES:
Cc1nnc2C(CC(N)=O)N=C(c3c(C)c(C)sc3-n12)c1ccc(Cl)cc1
Target:
Epigenetic Reader Domain

References

1. Devaiah BN, et al. Proc Natl Acad Sci U S A. 2012, 109(18), 6927-6932. 2. Moros A, et al. Leukemia. 2014. doi: 10.1038/leu.2014.106.