TargetMol

NSC-639829

Product Code:
 
TAR-T24553
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T24553-5mg5mg£850.00
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TAR-T24553-50mg50mg£1,661.00
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Quantity:
TAR-T24553-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
NSC-639829 is a tubulin polymerization inhibitor that acts by demonstrating potent antitumor activities against several cancer cell lines.
CAS:
134742-19-1
Formula:
C21H20BrN5O3
Molecular Weight:
470.327
Purity:
0.98
SMILES:
CN(C)c1ccccc1C(=O)NC(=O)Nc1ccc(Oc2ncc(Br)cn2)c(C)c1

References

1. Balcer-Kubiczek EK, Attarpour M, Edelman MJ. The synergistic effect of dimethylamino benzoylphenylurea (NSC #639829) and X-irradiation on human lung carcinoma cell lines. Cancer Chemother Pharmacol. 2007 May;59(6):781-7. Epub 2006 Sep 7. PubMed PMID: 16957930. 2. Rao VM, Nerurkar M, Pinnamaneni S, Rinaldi F, Raghavan K. Co-solubilization of poorly soluble drugs by micellization and complexation. Int J Pharm. 2006 Aug 17;319(1-2):98-106. Epub 2006 Apr 7. PubMed PMID: 16765542. 3. Hallur G, Jimeno A, Dalrymple S, Zhu T, Jung MK, Hidalgo M, Isaacs JT, Sukumar S, Hamel E, Khan SR. Benzoylphenylurea sulfur analogues with potent antitumor activity. J Med Chem. 2006 Apr 6;49(7):2357-60. PubMed PMID: 16570932. 4. Jain A, Sanghvi T, Yalkowsky SH. Liposome formulation of NSC-639829 using halothane as a solvent: a technical note. AAPS PharmSciTech. 2003 Oct 15;4(4):E52. PubMed PMID: 15198547; PubMed Central PMCID: PMC2750645.