Boc-ypgflt(O-tbu)

Product Code:

TAR-T25168

Product Group:

Inhibitors and Activators

Supplier:

TargetMol

Regulatory Status:

RUO

Shipping:

cool pack

Storage:

-20℃

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Code	Size	Price

TAR-T25168-5mg

5mg

£850.00

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Quantity:

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Further Information

Bioactivity:

Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.

CAS:

179124-36-8

Formula:

C44H64N6O11

Molecular Weight:

853.027

Purity:

0.98

SMILES:

CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H]([C@@H](C)OC(C)(C)C)C(O)=O

Documents

References

1. R?nai AZ, Magyar A, Orosz G, Borsodi A, Benyhe S, T?th G, Mak? E, K?tay E, Babka E, Medzihradszky K. Opioid antagonist properties of the highly delta-receptor-selective BOC-Tyr-Pro-Gly-Phe-Leu-Thr (OtBu) peptide and of its Phe1 and Mel1 analogues. Arch Int Pharmacodyn Ther. 1995 Nov-Dec;330(3):361-9. PubMed PMID: 8836454. 2. Mak? E, R?nai AZ, Ad?m G, Juh?sz G, Ritter L, Lest?r B, Crunelli V. Modulation by GABA(B) and delta opioid receptors of neurally induced responses in isolated guinea-pig taenia coli and human colonic circular muscle. J Physiol Paris. 2000 Mar-Apr;94(2):135-8. PubMed PMID: 10791695.