TargetMol

Fluperamide

Product Code:
 
TAR-T25430
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25430-5mg5mg£850.00
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TAR-T25430-50mg50mg£1,661.00
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Quantity:
TAR-T25430-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
Fluperamide is an antidiarrheal.
CAS:
53179-10-5
Formula:
C30H32ClF3N2O2
Molecular Weight:
545.04
Purity:
0.98
SMILES:
CN(C)C(=O)C(CCN1CCC(O)(CC1)c1ccc(Cl)c(c1)C(F)(F)F)(c1ccccc1)c1ccccc1

References

1. Megens AA, Canters LL, Awouters FH, Niemegeers CJ. Normalization of small intestinal propulsion with loperamide-like antidiarrheals in rats. Eur J Pharmacol. 1990 Mar 27;178(3):357-64. PubMed PMID: 2340864. 2. Reynolds IJ, Gould RJ, Snyder SH. Loperamide: blockade of calcium channels as a mechanism for antidiarrheal effects. J Pharmacol Exp Ther. 1984 Dec;231(3):628-32. PubMed PMID: 6502516. 3. Farrington H, Mendelsohn F, Chan S, Reinlib L, Guggino SE. Strychnine-binding proteins in intestinal cells: novel brucine binding site with binding affinities for alkaloids. J Pharmacol Exp Ther. 1994 Nov;271(2):1074-9. PubMed PMID: 7525935.