TargetMol

GR 100679

Product Code:
 
TAR-T25459
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25459-5mg5mg£850.00
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Quantity:
TAR-T25459-50mg50mg£1,661.00
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Quantity:
TAR-T25459-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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  • Further Information
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Further Information

Bioactivity:
GR 100679 is an antagonist of NK2 receptor.
CAS:
150351-87-4
Formula:
C34H44N6O5
Molecular Weight:
616.763
Purity:
0.98
SMILES:
C[C@H](NC(=O)CNC(=O)C1CCCCC1)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)NC(=O)[C@H](Cc1ccccc1)N(C)C

References

1. Stratton SC, Beresford IJ, Harvey FJ, Turpin MP, Hagan RM, Tyers MB. Anxiolytic activity of tachykinin NK2 receptor antagonists in the mouse light-dark box. Eur J Pharmacol. 1993 Dec 21;250(3):R11-2. PubMed PMID: 7906655. 2. Beresford IJ, Sheldrick RL, Ball DI, Turpin MP, Walsh DM, Hawcock AB, Coleman RA, Hagan RM, Tyers MB. GR159897, a potent non-peptide antagonist at tachykinin NK2 receptors. Eur J Pharmacol. 1995 Jan 16;272(2-3):241-8. PubMed PMID: 7713168. 3. Lundstrom K, Mills A, Allet E, Ceszkowski K, Agudo G, Chollet A, Liljestrom P. High-level expression of G protein-coupled receptors with the aid of the Semliki Forest virus expression system. J Recept Signal Transduct Res. 1995 Jan-Mar;15(1-4):23-32. PubMed PMID: 8903928. 4. Hagan RM, Beresford IJ, Stables J, Dupere J, Stubbs CM, Elliott PJ, Sheldrick RL, Chollet A, Kawashima E, McElroy AB, et al. Characterisation, CNS distribution and function of NK2 receptors studied using potent NK2 receptor antagonists. Regul Pept. 1993 Jul 2;46(1-2):9-19. PubMed PMID: 8210508.