TargetMol

GSK-A

Product Code:
 
TAR-T25471
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T25471-5mg5mg£1,010.00
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Quantity:
TAR-T25471-50mg50mg£1,982.00
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Quantity:
TAR-T25471-100mg100mg£2,560.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK-A is a Histone Lysine Methyltransferase EZH2 inhibitor.
CAS:
923894-97-7
Formula:
C21H25N5O2
Molecular Weight:
379.464
Purity:
0.98
SMILES:
CC(C)n1ncc2c(cc(nc12)C1CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O

References

1. Fraley KJ, Abberley L, Hottenstein CS, Ulicne JJ, Citerone DR, Szapacs ME. The Gyrolab? immunoassay system: a platform for automated bioanalysis and rapid sample turnaround. Bioanalysis. 2013 Jul;5(14):1765-74. doi: 10.4155/bio.13.145. PubMed PMID: 23862708. 2. Cheng Z, Zhang J, Liu H, Li Y, Zhao Y, Yang E. Central nervous system penetration for small molecule therapeutic agents does not increase in multiple sclerosis- and Alzheimer's disease-related animal models despite reported blood-brain barrier disruption. Drug Metab Dispos. 2010 Aug;38(8):1355-61. doi: 10.1124/dmd.110.033324. Epub 2010 Apr 28. PubMed PMID: 20427691. 3. Fries HE, Aiello M, Evans CA. Use of a variably sensitive selected reaction monitoring method to extend the linear dynamic range for quantitative high-performance liquid chromatography/tandem mass spectrometry. Rapid Commun Mass Spectrom. 2007;21(3):369-74. PubMed PMID: 17206741.