TargetMol

TRC210258

Product Code:
 
TAR-T26289
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26289-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T26289-50mg50mg£1,661.00
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Quantity:
TAR-T26289-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
TRC210258 is a TGR5 agonist that acts by decreasing glycemic and dyslipidemic cardiovascular risk in animal models of diabesity.
CAS:
1431553-15-9
Formula:
C20H14ClFN4O2
Molecular Weight:
396.81
Purity:
0.98
SMILES:
CN(C(=O)c1c(Oc2ccc(F)cc2)nc2ncccn12)c1ccc(Cl)cc1

References

1. Zambad SP, Tuli D, Mathur A, Ghalsasi SA, Chaudhary AR, Deshpande S, Gupta RC, Chauthaiwale V, Dutt C. TRC210258, a novel TGR5 agonist, reduces glycemic and dyslipidemic cardiovascular risk in animal models of diabesity. Diabetes Metab Syndr Obes. 2013 Dec 21;7:1-14. doi: 10.2147/DMSO.S50209. eCollection 2013. PubMed PMID: 24379686; PubMed Central PMCID: PMC3873233.