TargetMol

ACT-387042

Product Code:
 
TAR-T26558
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26558-5mg5mg£2,054.00
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Quantity:
TAR-T26558-50mg50mg£4,070.00
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Quantity:
TAR-T26558-100mg100mg£5,693.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
ACT-387042 is a Bacterial Topoisomerase Inhibitor, it has broad-spectrum activity against Gram-positive and Gram-negative bacteria.
CAS:
1229514-11-7
Formula:
C23H26FN5O4S
Molecular Weight:
487.55
Purity:
0.98
SMILES:
COc1ccc2ncc(F)c(C[C@H](O)[C@@H]3CC[C@H](CO3)NCc3cc4SCCOc4nn3)c2n1

References

1. Lepak AJ, Seiler P, Surivet JP, Ritz D, Kohl C, Andes DR. In Vivo Pharmacodynamic Target Investigation of Two Bacterial Topoisomerase Inhibitors, ACT-387042 and ACT-292706, in the Neutropenic Murine Thigh Model against Streptococcus pneumoniae and Staphylococcus aureus. Antimicrob Agents Chemother. 2016 May 23;60(6):3626-32. doi: 10.1128/AAC.00363-16. Print 2016 Jun. PubMed PMID: 27044547; PubMed Central PMCID: PMC4879394.