TargetMol

AP-521 (Free base)

Product Code:
 
TAR-T26640
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

No additional charges, what you see is what you pay! *

CodeSizePrice
TAR-T26640-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T26640-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T26640-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
Prices exclude any Taxes / VAT
Stay in control of your spending. These prices have no additional charges, not even shipping!
* Rare exceptions are clearly labelled (only 0.14% of items!).
Multibuy discounts available! Contact us to find what you can save.
This product comes from: United States.
Typical lead time: 10-14 working days.
Contact us for more accurate information.
  • Further Information
  • Documents
  • References
  • Show All

Further Information

Bioactivity:
AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.
CAS:
151227-58-6
Formula:
C20H19N3O3S
Molecular Weight:
381.45
Purity:
0.98
SMILES:
COc1ccc(cc1OC)C(=O)NC(=S)Nc1cccc2nc(C)ccc12

References

1. Kasahara K, Hashimoto S, Hattori T, Kawasaki K, Tsujita R, Nakazono O, Takao K, Kawakubo H, Nagatani T. The effects of AP521, a novel anxiolytic drug, in three anxiety models and on serotonergic neural transmission in rats. J Pharmacol Sci. 2015 Jan;127(1):109-16. doi: 10.1016/j.jphs.2014.11.008. PubMed PMID: 25704026.