TargetMol

BKM1644

Product Code:
 
TAR-T26831
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26831-5mg5mg£850.00
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This product comes from: United States.
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Further Information

Bioactivity:
BKM1644 is an effective inhibition of the proliferation of metastatic, castration-resistant PCa (mCRPC) cells.
CAS:
1070966-96-9
Formula:
C34H37Cl2F5N2O9P2
Molecular Weight:
845.51
Purity:
0.98
SMILES:
CCOP(=O)(OCC)C(NC(=O)[C@@H](Cc1ccc(OCc2c(Cl)cccc2Cl)cc1)NC(=O)C=Cc1c(F)c(F)c(F)c(F)c1F)P(=O)(OCC)OCC

References

1. Zhang S, Gera L, Mamouni K, Li X, Chen Z, Kucuk O, Wu D. Inhibition of skeletal growth of human prostate cancer by the combination of docetaxel and BKM1644: an aminobisphosphonate derivative. Oncotarget. 2016 May 10;7(19):27489-98. doi: 10.18632/oncotarget.8481. PubMed PMID: 27050371; PubMed Central PMCID: PMC5053666.