TargetMol

BL-1020 Mesylate

Product Code:
 
TAR-T26834
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26834-5mg5mg£850.00
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TAR-T26834-50mg50mg£1,661.00
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TAR-T26834-100mg100mg£2,079.00
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Further Information

Bioactivity:
BL-1020 is a GABA A receptor agonist and dopamine receptor antagonist. BL-1020 is an ester of GABA and perphenazine, and pharmacologically it acts as a GABA agonist and D2 antagonist. BL-1020 has shown pro-cognitive effects in the trials.
CAS:
916898-61-8
Formula:
C26H37ClN4O5S2
Molecular Weight:
585.18
Purity:
0.98
SMILES:
CS(O)(=O)=O.NCCCC(=O)OCCN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc23)CC1

References

1. Thyme S, Song Y. Computational Design of DNA-Binding Proteins. Methods Mol Biol. 2016;1414:265-83. doi: 10.1007/978-1-4939-3569-7_16. PubMed PMID: 27094297. 2. Geffen Y, Keefe R, Rabinowitz J, Anand R, Davidson M. Bl-1020, a new ?-aminobutyric acid-enhanced antipsychotic: results of 6-week, randomized, double-blind, controlled, efficacy and safety study. J Clin Psychiatry. 2012 Sep;73(9):e1168-74. doi: 10.4088/JCP.12m07642. PubMed PMID: 23059159. 3. Anand R, Geffen Y, Vasile D, Dan I. An open-label tolerability study of BL-1020 antipsychotic: a novel gamma aminobutyric acid ester of perphenazine. Clin Neuropharmacol. 2010 Nov-Dec;33(6):297-302. doi: 10.1097/WNF.0b013e3181f8d501. PubMed PMID: 20921890. 4. Fitzgerald PB. BL-1020, an oral antipsychotic agent that reduces dopamine activity and enhances GABAA activity, for the treatment of schizophrenia. Curr Opin Investig Drugs. 2010 Jan;11(1):92-100. Review. PubMed PMID: 20047163.