TargetMol

BMS-764459

Product Code:
 
TAR-T26856
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T26856-5mg5mg£1,171.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T26856-50mg50mg£2,303.00
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Quantity:
TAR-T26856-100mg100mg£3,042.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
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Further Information

Bioactivity:
BMS-764459 is a potent antagonist of corticotropin-releasing factor/hormone receptor 1 (CRHR-1).
CAS:
1188407-45-5
Formula:
C19H21F2N5O3
Molecular Weight:
405.406
Purity:
0.98
SMILES:
COC[C@H](C1CC1)n1cc(nc(Nc2cc(C)c(OC(F)F)nc2C)c1=O)C#N

References

1. Simic D, Euler C, Haines E, He A, Peden WM, Bunch RT, Sanderson T, Van Vleet T. MicroRNA changes associated with atypical CYP1A1 inducer BMS-764459. Toxicology. 2013 Sep 15;311(3):169-77. doi: 10.1016/j.tox.2013.06.006. Epub 2013 Jul 2. PubMed PMID: 23831372. 2. Gater D, Macauley D. American Chemical Society--238th National Meeting & Exposition. Developments in medicinal chemistry: part 2. 16-20 August 2009, Washington DC, USA. IDrugs. 2009 Oct;12(10):608-11. PubMed PMID: 19790005.