TargetMol

BMS-767778

Product Code:
 
TAR-T26857
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T26857-5mg5mg£1,572.00
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TAR-T26857-50mg50mg£3,107.00
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Quantity:
TAR-T26857-100mg100mg£4,247.00
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This product comes from: United States.
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Further Information

Bioactivity:
BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.
CAS:
915729-95-2
Formula:
C19H20Cl2N4O2
Molecular Weight:
407.3
Purity:
0.98
SMILES:
CN(C)C(=O)CN1Cc2nc(C)c(CN)c(c2C1=O)-c1ccc(Cl)cc1Cl

References

1. Devasthale P, Wang Y, Wang W, Fevig J, Feng J, Wang A, Harrity T, Egan D, Morgan N, Cap M, Fura A, Klei HE, Kish K, Weigelt C, Sun L, Levesque P, Moulin F, Li YX, Zahler R, Kirby MS, Hamann LG. Optimization of activity, selectivity, and liability profiles in 5-oxopyrrolopyridine DPP4 inhibitors leading to clinical candidate (Sa)-2-(3-(aminomethyl)-4-(2,4-dichlorophenyl)-2-methyl-5-oxo-5H-pyrrolo[3,4-b]py ridin-6(7H)-yl)-N,N-dimethylacetamide (BMS-767778). J Med Chem. 2013 Sep 26;56(18):7343-57. doi: 10.1021/jm4008906. PubMed PMID: 23964740.