TargetMol

Dasolampanel etibutil

Product Code:
 
TAR-T27123
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27123-5mg5mg£1,091.00
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TAR-T27123-50mg50mg£2,143.00
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TAR-T27123-100mg100mg£2,801.00
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Further Information

Bioactivity:
Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).
CAS:
503291-52-9
Formula:
C23H32ClN5O3
Molecular Weight:
461.99
Purity:
0.98
SMILES:
[H][C@@]12CC[C@@H](C[C@]1([H])C[C@H](NC2)C(=O)OCC(CC)CC)Oc1cccc(Cl)c1-c1nnn[nH]1

References

1. Petersen KL, Iyengar S, Chappell AS, Lobo ED, Reda H, Prucka WR, Verfaille SJ. Safety, tolerability, pharmacokinetics, and effects on human experimental pain of the selective ionotropic glutamate receptor 5 (iGluR5) antagonist LY545694 in healthy volunteers. Pain. 2014 May;155(5):929-36. doi: 10.1016/j.pain.2014.01.019. Epub 2014 Jan 31. PubMed PMID: 24486883. 2. Martinez-Perez JA, Iyengar S, Shannon HE, Bleakman D, Alt A, Clawson DK, Arnold BM, Bell MG, Bleisch TJ, Casta?o AM, Del Prado M, Dominguez E, Escribano AM, Filla SA, Ho KH, Hudziak KJ, Jones CK, Mateo A, Mathes BM, Mattiuz EL, Ogden AM, Simmons RM, Stack DR, Stratford RE, Winter MA, Wu Z, Ornstein PL. GluK1 antagonists from 6-(tetrazolyl)phenyl decahydroisoquinoline derivatives: in vitro profile and in vivo analgesic efficacy. Bioorg Med Chem Lett. 2013 Dec 1;23(23):6463-6. doi: 10.1016/j.bmcl.2013.09.045. Epub 2013 Sep 24. PubMed PMID: 24140446.