TargetMol

DG026

Product Code:
 
TAR-T27160
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27160-5mg5mg£1,653.00
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TAR-T27160-50mg50mg£3,267.00
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Quantity:
TAR-T27160-100mg100mg£4,488.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
DG026 is a IRAP inhibitor. DG026 ables to selectively downregulate IRAP-dependent cross-presentation by dendritic cells but leave ERAP1-dependent cross-presentation unaffected.
CAS:
2035046-17-2
Formula:
C35H40N3O4P
Molecular Weight:
597.696
Purity:
0.98
SMILES:
N[C@@H](CCc1ccccc1)P(O)(=O)CC(CC(c1ccccc1)c1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O

References

1. Ligand-Induced Conformational Change of Insulin-Regulated Aminopeptidase: Insights on Catalytic Mechanism and Active Site Plasticity Anastasia Mpakali, Emmanuel Saridakis, Karl Harlos, Yuguang Zhao, Paraskevi Kokkala, Dimitris Georgiadis, Petros Giastas, Athanasios Papakyriakou, and Efstratios Stratikos Publication Date (Web): March 22, 2017 (Article) doi: 10.1021/acs.jmedchem.6b01890