TargetMol

Efletirizine

Product Code:
 
TAR-T27244
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27244-1mg1mg£227.00
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TAR-T27244-5mg5mg£416.00
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TAR-T27244-10mg10mg£581.00
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TAR-T27244-25mg25mg£863.00
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TAR-T27244-50mg50mg£1,163.00
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TAR-T27244-100mg100mg£1,540.00
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Quantity:
TAR-T27244-500mg500mg£3,026.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Efletirizine, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.
CAS:
150756-35-7
Formula:
C21H24F2N2O3
Molecular Weight:
390.431
Pathway:
Neuroscience|GPCR/G Protein|Metabolism|Immunology/Inflammation
Purity:
0.98
SMILES:
OC(=O)COCCN1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1
Target:
Histamine Receptor|Lipoxygenase

References

1. Lewis TA, Young MA, Arrington MP, Bayless L, Cai X, Collart P, Eckman JB, Ellis JL, Ene DG, Libertine L, Nicolas JM, Scannell RT, Wels BF, Wenberg K, Wypij DM. Cetirizine and loratadine-based antihistamines with 5-lipoxygenase inhibitory activity. Bioorg Med Chem Lett. 2004 Nov 15;14(22):5591-4. PubMed PMID: 15482930. 2. Salmun LM. Antihistamines in late-phase clinical development for allergic disease. Expert Opin Investig Drugs. 2002 Feb;11(2):259-73. Review. PubMed PMID: 11829715. 3. Coe RA, DeCesare LS, Lee JW. Quantitation of efletirizine in human plasma and urine using automated solid-phase extraction and column-switching high-performance liquid chromatography. J Chromatogr B Biomed Sci Appl. 1999 Jul 9;730(2):239-47. PubMed PMID: 10448959.